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sion in singleuse vials Improved activity against grampositive and atypical pathogens Investigational fluoroquinolones Moxifloxacin Improved activity against grampositive bacteria, atypical pathogens, and anaerobes Gatifloxacin Clinafloxacin Gemifloxacin Sitafloxacin 硝基呋喃類 Nitrofurans ? 呋喃妥因 nitrofurantoin 泌尿道抗菌藥 Urinary antiseptics ? 呋喃唑酮 furanzolidone (痢特靈) 腸道感染 —腸炎、菌痢 抗幽門(mén)螺桿菌 —胃潰瘍 硝基咪唑類 Nitromidazoles ? 甲硝唑 metronidazole 厭氧菌、混合性腹腔感染 細(xì)菌性或滴蟲(chóng)性陰道炎 抗幽門(mén)螺桿菌 —胃潰瘍 自學(xué)! 謝謝觀看 /歡迎下載 BY FAITH I MEAN A VISION OF GOOD ONE CHERISHES AND THE ENTHUSIASM THAT PUSHES ONE TO SEEK ITS FULFILLMENT REGARDLESS OF OBSTACLES. BY FAITH I BY FAITH 。 broad indications for systemic use Ofloxacin (Floxin) OrthoMcNeil Pharmaceuticals 200, 300, and 400mg tablets?;瘜W(xué)治療藥物 Chemotherapeutic Drugs 學(xué)習(xí)提要 掌握喹諾酮及磺胺類藥物的作用機(jī)制及區(qū)別點(diǎn) 掌握各組喹諾酮藥物的抗菌特性 掌握喹諾酮及磺胺類藥物的臨床應(yīng)用及常見(jiàn)不良反應(yīng)及產(chǎn)生耐藥機(jī)制 ? 化學(xué)治療藥物 Ideal: ?對(duì)細(xì)菌等病原微生物、寄生蟲(chóng)和癌細(xì)胞有選擇性殺滅作用 ?對(duì) Host無(wú)毒或輕度毒性 Note ? Host, Pathogen and Drugs ? Reasonable, Safety and Effective 治療指數(shù) =LD50/ED50 Certain Safety Factor 確實(shí)安全系數(shù) ? 化療指數(shù)越大則說(shuō)明藥物毒性越低 ? 治療指數(shù)大于 5,可做臨床研究 ? 治療效果越高? ? 化療指數(shù) Chemotherapeutic index Unsatisfactory of safety margin 不滿意的安